Cart
sales@molnova.com
Eletriptan hydrobromide
CAS No. 177834-92-3
Eletriptan hydrobromide( UK 116044 hydrobromide )
Catalog No. M12677 CAS No. 177834-92-3
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 54 | In Stock |
|
| 2MG | 31 | In Stock |
|
| 5MG | 49 | In Stock |
|
| 10MG | 61 | In Stock |
|
| 25MG | 129 | In Stock |
|
| 50MG | 212 | In Stock |
|
| 100MG | 352 | In Stock |
|
| 200MG | 520 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameEletriptan hydrobromide
-
NoteResearch use only, not for human use.
-
Brief DescriptionEletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
-
DescriptionEletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migrainev Approved.
-
In Vitro——
-
In Vivo——
-
SynonymsUK 116044 hydrobromide
-
PathwayGPCR/G Protein
-
Target5-HT Receptor
-
Recptor5-HT1B|5-HT1D
-
Research AreaNeurological Disease
-
IndicationMigraine
Chemical Information
-
CAS Number177834-92-3
-
Formula Weight463.43
-
Molecular FormulaC22H26N2O2S.HBr
-
Purity>98% (HPLC)
-
SolubilityDMSO: 46.3 mg/mL (100 mM) （ < 1 mg/ml refers to the product slightly soluble or insoluble )
-
SMILESCN1CCC[C@@H]1CC2=CNC3=C2C=C(C=C3)CCS(=O)(=O)C4=CC=CC=C4.Br
-
Chemical Name3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
molnova catalog
related products
-
SB228357
SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.
-
SB 216641
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety and depression.
-
SUVN-502 mesylate hy...
SUVN-502 (SUVN502)?is a?potent, selective, brain penetrant and orally active 5-HT6 receptor antagonist with Ki of 2.04 nM.
