DDR inhibitor X

CAS No. 1644069-80-6

DDR inhibitor X( —— )

Catalog No. M12505 CAS No. 1644069-80-6

DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 372 Get Quote
10MG 597 Get Quote
25MG 1197 Get Quote
50MG 1908 Get Quote
100MG 2583 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    DDR inhibitor X
  • Note
    Research use only, not for human use.
  • Brief Description
    DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2.
  • Description
    DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
  • In Vitro
    DDR Inhibitor (Example 6) is a potent DDR inhibitor, with an IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Tyrosine Kinase
  • Target
    DDR
  • Recptor
    DDR
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1644069-80-6
  • Formula Weight
    417.444
  • Molecular Formula
    C23H20FN5O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 65 mg/mL 155.71 mM; H2O : < 0.1 mg/mL
  • SMILES
    CC1=C(C=C(C=C1)CNC(=O)NC2=CC(=CC=C2)F)NC(=O)C3=CN=C4N3C=CC=C4
  • Chemical Name
    N-[5-[[[(3-Fluorophenyl)carbamoyl]amino]methyl]-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Patent WO2015004481A1.
molnova catalog
related products
  • DDR2-IN-5

    DDR2-IN-5 is a potent, dual DDR2/SRC inhibitor with IC50 of 56/12 nM.

  • DDR1 inhibitor 7rh

    DDR1 inhibitor 7rh is a potent, selective, ATP-competitive, orally available Discoidin domain receptor 1 (DDR1) inhibitor with IC50 of 6.8 nM in cell-free kinase assays.

  • LCB 03-0110 dihydroc...

    LCB 03-0110 is a potent, ATP-competitive inhibitor of Discoidin domain receptor (DDR) family and c-Src tyrosine kinase family.