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DDR inhibitor X
CAS No. 1644069-80-6
DDR inhibitor X( —— )
Catalog No. M12505 CAS No. 1644069-80-6
DDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 259 | In Stock |
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| 5MG | 235 | In Stock |
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| 10MG | 377 | In Stock |
|
| 25MG | 758 | In Stock |
|
| 50MG | 1181 | In Stock |
|
| 100MG | 1600 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDDR inhibitor X
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NoteResearch use only, not for human use.
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Brief DescriptionDDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2.
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DescriptionDDR inhibitor X is a potent discoidin domain receptor (DDR) inhibitor with IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
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In VitroDDR Inhibitor (Example 6) is a potent DDR inhibitor, with an IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM.
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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TargetDDR
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RecptorDDR
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1644069-80-6
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Formula Weight417.444
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Molecular FormulaC23H20FN5O2
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Purity>98% (HPLC)
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SolubilityDMSO : 65 mg/mL 155.71 mM; H2O : < 0.1 mg/mL
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SMILESCC1=C(C=C(C=C1)CNC(=O)NC2=CC(=CC=C2)F)NC(=O)C3=CN=C4N3C=CC=C4
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Chemical NameN-[5-[[[(3-Fluorophenyl)carbamoyl]amino]methyl]-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Patent WO2015004481A1.
molnova catalog
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