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Bosentan Hydrate
CAS No. 157212-55-0
Bosentan Hydrate( —— )
Catalog No. M12244 CAS No. 157212-55-0
Bosentan is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 35 | In Stock |
|
| 50MG | 50 | In Stock |
|
| 100MG | 87 | In Stock |
|
| 200MG | 147 | In Stock |
|
| 500MG | 267 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBosentan Hydrate
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NoteResearch use only, not for human use.
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Brief DescriptionBosentan is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.
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DescriptionBosentan is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetEndothelin Receptor
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RecptorET-B| ET-A
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number157212-55-0
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Formula Weight569.63
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Molecular FormulaC??H??N?O?S
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Purity>98% (HPLC)
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SolubilityDMSO:93 mg/mL (163.3 mM);Ethanol:2 mg/mL (3.51 mM);Water:<1 mg/Ml
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SMILESO.COC1=CC=CC=C1OC1=C(OCCO)N=C(N=C1NS(=O)(=O)C1=CC=C(C=C1)C(C)(C)C)C1=NC=CC=N1 |c:4,6,10,16,18,27,29,38,40,t:2,25,36|
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Clozel M, et al. J Pharmacol Exp Ther, 1994, 270(1), 228-235.
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