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Ischemin
CAS No. 1357059-00-7
Ischemin( —— )
Catalog No. M11461 CAS No. 1357059-00-7
A cell permeable CBP bromodomain inhibitor with Kd of 19 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameIschemin
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NoteResearch use only, not for human use.
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Brief DescriptionA cell permeable CBP bromodomain inhibitor with Kd of 19 uM.
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DescriptionA cell permeable CBP bromodomain inhibitor with Kd of 19 uM; inhibits the acetyl-lysine binding activity of CBP, inhibits p53 interaction with CBP and decreases p53 transcriptional activity; protects against doxorubicin-induced apoptosis in cardiomyocytes in vitro.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research Area——
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Indication——
Chemical Information
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CAS Number1357059-00-7
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Formula Weight335.378
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Molecular FormulaC15H17N3O4S
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1=CC(=C(C=C1N=NC2=C(C=C(C(=C2)C)O)N)S(=O)(=O)O)C
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Chemical Name5-[(1E)-2-(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-2,4-dimethylbenzenesulfonic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Borah JC, et al. Chem Biol. 2011 Apr 22;18(4):531-41.
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