SB-699393
CAS No. 1348166-93-7
SB-699393( SB699393 )
Catalog No. M11412 CAS No. 1348166-93-7
SB-699393 is a potent, selective and CNS penetrant B-Raf inhibitor with Kd of 7.2 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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Biological Information
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Product NameSB-699393
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NoteResearch use only, not for human use.
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Brief DescriptionSB-699393 is a potent, selective and CNS penetrant B-Raf inhibitor with Kd of 7.2 nM.
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DescriptionSB-699393 is a potent, selective and CNS penetrant B-Raf inhibitor with Kd of 7.2 nM; possesses enhanced CNS penetration (BB ratio=0.8:1) compared with SB-590885.
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In Vitro——
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In Vivo——
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SynonymsSB699393
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PathwayMAPK/ERK Signaling
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TargetRaf
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RecptorRaf
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Research Area——
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Indication——
Chemical Information
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CAS Number1348166-93-7
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Formula Weight403.482
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Molecular FormulaC24H25N3O3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(E)-((5-(5-(morpholinomethyl)-2-(pyridin-4-yl)furan-3-yl)-2,3-dihydro-1H-inden-1-ylidene)amino)methanol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Takle AK, et al. Bioorg Med Chem Lett. 2008 Aug 1;18(15):4373-6.
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