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PF-2545920

CAS No. 1292799-56-4

PF-2545920( —— )

Catalog No. M11184 CAS No. 1292799-56-4

PF-2545920 is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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5MG	182	In Stock
10MG	251	In Stock
25MG	410	In Stock
50MG	602	In Stock
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Biological Information

Product Name

PF-2545920
Note

Research use only, not for human use.
Brief Description

PF-2545920 is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM.
Description

PF-2545920 is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM, with >1000-fold selectivity over the PDE.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Angiogenesis
Target

PDE
Recptor

PDE10A
Research Area

——
Indication

——

Chemical Information

CAS Number

1292799-56-4
Formula Weight

392.45
Molecular Formula

C25H20N4O
Purity

>98% (HPLC)
Solubility

Ethanol: 79 mg/mL (201.29 mM); DMSO: 79 mg/mL (201.29 mM)
SMILES

CN1C=C(C(=N1)C2=CC=C(C=C2)OCC3=NC4=CC=CC=C4C=C3)C5=CC=NC=C5
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Wilson JM, et al. Neuropharmacology. 2015 Dec;99:379-86.

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