LGD-4033( LGD 4033 | LGD4033 | VK-5211 )

Catalog No. M10567 CAS No. 1165910-22-4

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HNMR

HPLC

MSDS

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Product Name

LGD-4033
Note

Research use only, not for human use.
Brief Description

A novel nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity.
Description

A novel nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity; has favorable pharmacokinetic profile, and increases lean body mass even during this short period without change in prostate-specific antigen.Other Indication Phase 2 Clinical.
In Vitro

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In Vivo

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Synonyms

LGD 4033 | LGD4033 | VK-5211
Pathway

Endocrinology/Hormones
Target

Androgen Receptor (AR)
Recptor

Androgen Receptor (AR)
Research Area

Other Indications
Indication

Other Disease

CAS Number

1165910-22-4
Formula Weight

338.25
Molecular Formula

C14H12F6N2O
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : ≥ 100 mg/mL (295.64 mM)
SMILES

N#CC1=CC=C(N2[C@@H]([C@@H](O)C(F)(F)F)CCC2)C=C1C(F)(F)F
Chemical Name

4-((R)-2-((R)-2,2,2-trifluoro-1-hydroxyethyl)pyrrolidin-1-yl)-2-(trifluoromethyl)benzonitrile

1. Basaria S, et al. J Gerontol A Biol Sci Med Sci. 2013 Jan;68(1):87-95.

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