CP-466722

CAS No. 1080622-86-1

CP-466722( CP466722 | CP 466722 )

Catalog No. M10322 CAS No. 1080622-86-1

A poten and selective ATM inhibitor without effect on ATR kinase; does not inhibit PI3K, PI3K-like protein kinases or Abl kinase and disrupts ATM-dependent cell cycle checkpoints in cells.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 40 In Stock
5MG 61 In Stock
10MG 105 In Stock
25MG 174 In Stock
50MG 281 In Stock
100MG 455 In Stock
500MG 1017 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CP-466722
  • Note
    Research use only, not for human use.
  • Brief Description
    A poten and selective ATM inhibitor without effect on ATR kinase; does not inhibit PI3K, PI3K-like protein kinases or Abl kinase and disrupts ATM-dependent cell cycle checkpoints in cells.
  • Description
    A poten and selective ATM inhibitor without effect on ATR kinase; does not inhibit PI3K, PI3K-like protein kinases or Abl kinase and disrupts ATM-dependent cell cycle checkpoints in cells.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CP466722 | CP 466722
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    ATM/ATR
  • Recptor
    ATM
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1080622-86-1
  • Formula Weight
    349.3467
  • Molecular Formula
    C17H15N7O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 7 mg/mL (Need warming)
  • SMILES
    COC1=C(C=C2C(=C1)C(=NC=N2)N3C(=NC(=N3)C4=CC=CC=N4)N)OC
  • Chemical Name
    1H-1,2,4-Triazol-5-amine, 1-(6,7-dimethoxy-4-quinazolinyl)-3-(2-pyridinyl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Rainey MD, et al. Cancer Res. 2008 Sep 15;68(18):7466-74.
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