PK-14105( PK14105 )

Catalog No. M10296 CAS No. 107257-28-3

A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

PK-14105
Note

Research use only, not for human use.
Brief Description

A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.
Description

A potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM; attaches covalently and specifically to all the PBS when cardiac membranes are irradiated with this compound under ultraviolet light.
In Vitro

——
In Vivo

——
Synonyms

PK14105
Pathway

Membrane Transporter/Ion Channel
Target

GAT
Recptor

GAT
Research Area

Other Indications
Indication

——

Chemical Information

CAS Number

107257-28-3
Formula Weight

381.4002
Molecular Formula

C21H20FN3O3
Purity

>98% (HPLC)
Solubility

DMSO: ≥ 30 mg/mL
SMILES

O=C(C1=CC2=C(C(C3=CC([N+]([O-])=O)=CC=C3F)=N1)C=CC=C2)N(C(CC)C)C
Chemical Name

3-Isoquinolinecarboxamide, 1-(2-fluoro-5-nitrophenyl)-N-methyl-N-(1-methylpropyl)-

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Doble A, et al. Mol Pharmacol. 1987 Jan;31(1):42-9. 2. Doble A, et al. J Recept Res. 1987;7(1-4):55-70. 3. Skowroński R, et al. Eur J Pharmacol. 1988 Mar 29;148(2):187-93.

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