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KJ-Pyr-9
CAS No. 581073-80-5
KJ-Pyr-9( KJ Pyr9 )
Catalog No. M15131 CAS No. 581073-80-5
KJ-Pyr-9 is a novel small-molecule inhibitor of c-Myc (Kd=6.5 ± 1.0 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 30 | Get Quote |
|
| 5MG | 47 | Get Quote |
|
| 10MG | 67 | Get Quote |
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| 25MG | 133 | Get Quote |
|
| 50MG | 264 | Get Quote |
|
| 100MG | 482 | Get Quote |
|
| 200MG | 647 | Get Quote |
|
| 500MG | 1008 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameKJ-Pyr-9
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NoteResearch use only, not for human use.
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Brief DescriptionKJ-Pyr-9 is a novel small-molecule inhibitor of c-Myc (Kd=6.5 ± 1.0 nM).
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DescriptionKJ-Pyr-9 is a novel small-molecule inhibitor of c-Myc (Kd=6.5 ± 1.0 nM); interferes with MYC-MAX complex formation and inhibits MYC-induced oncogenic transformation in cells; active in xenograft mice.
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In Vitro——
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In Vivo——
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SynonymsKJ Pyr9
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PathwayCell Cycle/DNA Damage
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Targetc-Myc
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Recptorc-Myc
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number581073-80-5
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Formula Weight385.3722
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Molecular FormulaC22H15N3O4
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(N)C1=CC=C(C2=CC(C3=CC=CO3)=NC(C4=CC=C([N+]([O-])=O)C=C4)=C2)C=C1
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Chemical NameBenzamide, 4-[2-(2-furanyl)-6-(4-nitrophenyl)-4-pyridinyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hart JR, et al. Proc Natl Acad Sci U S A. 2014 Aug 26;111(34):12556-61.
2. Raffeiner P, et al. Oncotarget. 2014 Oct 15;5(19):8869-78.
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