H2L5186303

CAS No. 139262-76-3

H2L5186303( ZINC33388081 )

Catalog No. M27634 CAS No. 139262-76-3

H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 88 Get Quote
10MG 160 Get Quote
25MG 357 Get Quote
50MG 530 Get Quote
100MG 759 Get Quote
500MG 1557 Get Quote
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Biological Information

  • Product Name
    H2L5186303
  • Note
    Research use only, not for human use.
  • Brief Description
    H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.
  • Description
    H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.(In Vitro):The high cell invasion activity of HT1080-M6 cells is significantly suppressed by H2L5186303.(In Vivo):H2L5186303 shows strong suppressive efficacy when administered before OVA sensitization and challenge, such as suppression of airway hyper responsiveness, inflammatory cytokine levels, mucin production, and eosinophil numbers.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ZINC33388081
  • Pathway
    GPCR/G Protein
  • Target
    LPA Receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    139262-76-3
  • Formula Weight
    488.45
  • Molecular Formula
    C26H20N2O8
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (511.82 mM)
  • SMILES
    O(C1=CC(OC2=CC=C(NC(/C=C\C(O)=O)=O)C=C2)=CC=C1)C3=CC=C(NC(/C=C\C(O)=O)=O)C=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Gibson Francis S. Synthesis of paclitaxel by protecting the 7-?hydroxyl of baccatin III using a strong base and an electrophile. WO9945001A1.
molnova catalog
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