Cart
sales@molnova.com
GSK-812
CAS No. 630407-66-8
GSK-812( GSK812 )
Catalog No. M15383 CAS No. 630407-66-8
GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameGSK-812
-
NoteResearch use only, not for human use.
-
Brief DescriptionGSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
-
DescriptionGSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina, shows has polypharmacology antagonizing multiple receptors, including D2 and D3 receptors, and 5-HT2A, 2C, and 5-HT6 receptors.
-
In Vitro——
-
In Vivo——
-
SynonymsGSK812
-
PathwayEndocrinology/Hormones
-
Target5-HT Receptor
-
Recptor5-HT Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number630407-66-8
-
Formula Weight471.996
-
Molecular FormulaC25H26ClNO4S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCN1CCC2=CC(=C(C=C2CC1)S(=O)(=O)C3=CC=C(C=C3)OCC4=CC=C(C=C4)Cl)OC
-
Chemical Name7-[4-(4-chloro-benzyloxy)-benzenesulfonyl]-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Baranov P, et al. J Ocul Pharmacol Ther. 2017 Jun;33(5):412-422.
molnova catalog
related products
-
Pindolol
Pindolol is a nonselective β-blocker with partial beta-adrenergic receptor agonist activity, also functions as a 5-HT1A receptor weak partial agonist / antagonist (Ki=33nM).
-
Pimavanserin
Pimavanserin(ACP-103) is a potent and selective 5-HT2A receptor inverse agonist with mean pIC50 of with 8.7 in the cell-based functional assay.
-
EMDT oxalate
EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.
