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DGY-06-116
CAS No. ——
DGY-06-116( —— )
Catalog No. M22645 CAS No. ——
DGY-06-116 is an selective and irreversible covalent inhibitor of Src and FGFR1 with IC50 value of 3nM and 8340 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 165 | In Stock |
|
| 5MG | 235 | In Stock |
|
| 10MG | 393 | In Stock |
|
| 25MG | 657 | In Stock |
|
| 50MG | 1007 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameDGY-06-116
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NoteResearch use only, not for human use.
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Brief DescriptionDGY-06-116 is an selective and irreversible covalent inhibitor of Src and FGFR1 with IC50 value of 3nM and 8340 nM, respectively.
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DescriptionDGY-06-116 is an selective and irreversible covalent inhibitor of Src and FGFR1 with IC50 value of 3nM and 8340 nM, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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TargetSrc
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RecptorSrc|FGFR1
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight597.11
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Molecular FormulaC32H33ClN8O2
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL (167.47 mM)
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SMILESCN1CCN(CC1)c1ccc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)c(Nc3ccccc3NC(=O)C=C)n2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Gurbani D , Du G , Henning N J , et al. Structure and Characterization of a Covalent Inhibitor of Src Kinase[J]. Frontiers in Molecular Bioences, 2020, 7:81.
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