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CS3
CAS No. 1207457-11-1
CS3( cIAP inhibitor CS3 )
Catalog No. M10766 CAS No. 1207457-11-1
CS3 is a potent, selective cIAP1 and cIAP2 inhibitor with IC50 of 16 nM and 85 nM respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameCS3
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NoteResearch use only, not for human use.
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Brief DescriptionCS3 is a potent, selective cIAP1 and cIAP2 inhibitor with IC50 of 16 nM and 85 nM respectively.
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DescriptionCS3 is a potent, selective cIAP1 and cIAP2 inhibitor with IC50 of 16 nM and 85 nM respectively, shows no significant activity against XIAP (IC50>34 uM).
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In Vitro——
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In Vivo——
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SynonymscIAP inhibitor CS3
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PathwayApoptosis
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TargetIAP
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RecptorIAP
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Research Area——
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Indication——
Chemical Information
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CAS Number1207457-11-1
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Formula Weight506.651
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Molecular FormulaC28H38N6O3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(2S,3S)-1-((S)-2-cyclohexyl-2-((S)-2-(methylamino)propanamido)acetyl)-3-methyl-N-(2-(pyrimidin-2-yl)phenyl)pyrrolidine-2-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ndubaku C, et al. ACS Chem Biol. 2009 Jul 17;4(7):557-66.
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