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CAY10444

CAS No. 298186-80-8

CAY10444( —— )

Catalog No. M33970 CAS No. 298186-80-8

CAY10444 is an S1P3 specific antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 37 Get Quote
10MG 65 Get Quote
25MG 135 Get Quote
50MG 227 Get Quote
100MG 372 Get Quote
200MG 505 Get Quote
500MG 795 Get Quote
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Biological Information

  • Product Name
    CAY10444
  • Note
    Research use only, not for human use.
  • Brief Description
    CAY10444 is an S1P3 specific antagonist.
  • Description
    CAY10444 (BML-241) is a sphingosine-1-phosphate 3 (S1P3) antagonist. CAY10444 inhibits by 37% S1P-induced increases in Ca2+ in HeLa cells expressing S1P3 receptors.
  • In Vitro
    BML-241 inhibits increases in intracellular Ca2+ concentration via P2 receptor or α1A-adrenoceptor stimulation and α1A-adrenoceptor-mediated contraction of rat mesenteric artery, while it does not affect S1P3-mediated decrease of Forskolin-induced cyclic AMP accumulation.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    298186-80-8
  • Formula Weight
    287.46
  • Molecular Formula
    C15H29NO2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 41.67 mg/mL (144.96 mM; Ultrasonic (<80°C)
  • SMILES
    CCCCCCCCCCCC1N[C@@H](CS1)C(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Salvatore Salomone, et al. Selectivity and specificity of sphingosine-1-phosphate receptor ligands: caveats and critical thinking in characterizing receptor-mediated effects. Front Pharmacol. 2011 Feb 22;2:9. ?
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