CAY10444( —— )

Catalog No. M33970 CAS No. 298186-80-8

CAY10444 is an S1P3 specific antagonist.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

CAY10444
Note

Research use only, not for human use.
Brief Description

CAY10444 is an S1P3 specific antagonist.
Description

CAY10444 (BML-241) is a sphingosine-1-phosphate 3 (S1P3) antagonist. CAY10444 inhibits by 37% S1P-induced increases in Ca2+ in HeLa cells expressing S1P3 receptors.
In Vitro

BML-241 inhibits increases in intracellular Ca2+ concentration via P2 receptor or α1A-adrenoceptor stimulation and α1A-adrenoceptor-mediated contraction of rat mesenteric artery, while it does not affect S1P3-mediated decrease of Forskolin-induced cyclic AMP accumulation.
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Others
Research Area

——
Indication

——

Chemical Information

CAS Number

298186-80-8
Formula Weight

287.46
Molecular Formula

C15H29NO2S
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 41.67 mg/mL (144.96 mM; Ultrasonic (<80°C)
SMILES

CCCCCCCCCCCC1N[C@@H](CS1)C(O)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Salvatore Salomone, et al. Selectivity and specificity of sphingosine-1-phosphate receptor ligands: caveats and critical thinking in characterizing receptor-mediated effects. Front Pharmacol. 2011 Feb 22;2:9. ?

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