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BPDBA
CAS No. 312281-74-6
BPDBA( —— )
Catalog No. M34193 CAS No. 312281-74-6
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 53 | Get Quote |
|
| 10MG | 85 | Get Quote |
|
| 25MG | 170 | Get Quote |
|
| 50MG | 273 | Get Quote |
|
| 100MG | 431 | Get Quote |
|
| 500MG | 945 | Get Quote |
|
| 1G | 1251 | Get Quote |
|
Biological Information
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Product NameBPDBA
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NoteResearch use only, not for human use.
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Brief DescriptionBPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.
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DescriptionBPDBA is a selective and noncompetitive betaine/GABA transporter (BGT-1) inhibitor with IC50s of 20 μM and 35 μM against human BGT-1 and mouse GAT2, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGABA Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number312281-74-6
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Formula Weight363.28
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Molecular FormulaC19H20Cl2N2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (275.27 mM; Ultrasonic )
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SMILESC(N1CCC(NC(=O)C2=C(Cl)C=C(Cl)C=C2)CC1)C3=CC=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kragholm B, et al. Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile. Biochem Pharmacol. 2013 Aug 15;86(4):521-8.?
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