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BMS 830216
CAS No. 1197420-06-6
BMS 830216( BMS-830216 | BMS830216 )
Catalog No. M10704 CAS No. 1197420-06-6
The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 1053 | Get Quote |
|
| 50MG | 2142 | Get Quote |
|
| 100MG | 2790 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameBMS 830216
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NoteResearch use only, not for human use.
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Brief DescriptionThe the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
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DescriptionThe the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM; shows potential for treatment of obesity.ObesityPhase 2 Discontinued.
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In Vitro——
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In Vivo——
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SynonymsBMS-830216 | BMS830216
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PathwayGPCR/G Protein
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TargetMCHR
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RecptorMCHR
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Research AreaMetabolic Disease
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IndicationObesity
Chemical Information
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CAS Number1197420-06-6
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Formula Weight548.931
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Molecular FormulaC24H22ClN2O7PS
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Purity>98% (HPLC)
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Solubility——
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SMILESCOC1=C(C=CC(=C1)N2C=NC3=C(C2=O)SC(=C3)C4=CC=C(C=C4)Cl)OCC(C5CC5)OP(=O)(O)O
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Chemical Name(R)-2-(4-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimidin-3(4H)-yl)-2-methoxyphenoxy)-1-cyclopropylethyl dihydrogen phosphate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.
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BMS 830216
The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
