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Apatinib
CAS No. 811803-05-1
Apatinib( YN968D1 )
Catalog No. M16035 CAS No. 811803-05-1
Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 76 | In Stock |
|
| 5MG | 108 | In Stock |
|
| 10MG | 137 | In Stock |
|
| 25MG | 233 | In Stock |
|
| 50MG | 350 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameApatinib
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NoteResearch use only, not for human use.
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Brief DescriptionApatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
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DescriptionApatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
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In Vitro——
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In Vivo——
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SynonymsYN968D1
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PathwayAngiogenesis
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Targetc-Kit
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Recptorc-Kit| RET| c-Src| VEGFR2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number811803-05-1
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Formula Weight397.48
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Molecular FormulaC24H23N5O
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Purity>98% (HPLC)
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SolubilityDMSO: 22 mg/mL (44.57 mM)
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SMILESCS(O)(=O)=O.O=C(NC1=CC=C(C=C1)C1(CCCC1)C#N)C1=C(NCC2=CC=NC=C2)N=CC=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tian S, et al. Y Sci, 2011, 102(7), 1374-1380.
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