(1R,2R)-2-PCCA hydrochloride( —— )

Catalog No. M33183 CAS No. 1609563-71-4

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HNMR

HPLC

MSDS

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Product Name

(1R,2R)-2-PCCA hydrochloride
Note

Research use only, not for human use.
Brief Description

(1R,2R)-2-PCCA hydrochloride is a potent, selective, and blood-brain-barrier-crossing GPR88 receptor agonist with an EC50 value of 1140 n in striatal membranes of WT mice; it can be used to study the central nervous system.
Description

(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay.
In Vitro

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In Vivo

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Synonyms

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Pathway

Others
Target

Other Targets
Recptor

Others
Research Area

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Indication

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CAS Number

1609563-71-4
Formula Weight

528.56
Molecular Formula

C30H39Cl2N3O
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 50 mg/mL (94.60 mM; Ultrasonic )
SMILES

Cl.Cl.CCCc1ccc(cc1)-c1ccc(cc1)N(C[C@@H](N)[C@@H](C)CC)C(=O)[C@@H]1C[C@H]1c1ccccn1
Chemical Name

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1. Bi, Yingzhi, et al. Modulators of G Protein-Coupled Receptor 88. US 20110251204 A1.

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