Ro 31-8220 is a pan-PKC inhibitor for PKC-α/βI/βII/γ/ε (IC50: 5/24/14/27/24 nM), and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β.

[bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.

AICAR monophosphate, a purine precursor with antineoplastic activity, is important in the treatment of metabolic diseases such as type 2 diabetes as well as a possible treatment of various cancer types.