ML192

CAS No. 460331-61-7

ML192( —— )

Catalog No. M34655 CAS No. 460331-61-7

ML192 (CID1434953) is a selective GPR55 ligand antagonist. ML192 is an inhibitor that inhibits β-arrestin transport, ERK1/2 phosphorylation, and PKCβII translocation.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 70 Get Quote
5MG 107 Get Quote
10MG 178 Get Quote
25MG 293 Get Quote
50MG 423 Get Quote
100MG 583 Get Quote
500MG 1161 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    ML192
  • Note
    Research use only, not for human use.
  • Brief Description
    ML192 (CID1434953) is a selective GPR55 ligand antagonist. ML192 is an inhibitor that inhibits β-arrestin transport, ERK1/2 phosphorylation, and PKCβII translocation.
  • Description
    ML192 is a selective ligand antagonist of GPR55. ML192 inhibits the β-arrestin trafficking, ERK1/2 phosphorylation and PKCβII translocation.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Arrestin | Cannabinoid Receptor | GPR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    460331-61-7
  • Formula Weight
    382.48
  • Molecular Formula
    C20H22N4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (261.45 mM; Ultrasonic )
  • SMILES
    Cc1nc(N2CCN(CC2)C(=O)c2ccco2)c2c3CCCCc3sc2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kotsikorou E, et al. Identification of the GPR55 antagonist binding site using a novel set of high-potency GPR55 selective ligands. Biochemistry. 2013 Dec 31;52(52):9456-69.?
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