M1001

CAS No. 874590-32-6

M1001( —— )

Catalog No. M21074 CAS No. 874590-32-6

M1001 is a HIF-2α?agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 79 Get Quote
5MG 132 Get Quote
10MG 222 Get Quote
25MG 447 Get Quote
50MG 651 Get Quote
100MG 888 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    M1001
  • Note
    Research use only, not for human use.
  • Brief Description
    M1001 is a HIF-2α?agonist.
  • Description
    M1001 is a HIF-2α?agonist.
  • In Vitro
    Western Blot Analysis Cell Line:786-O cells Concentration:10?μM Incubation Time:Result:Increased the expression of HIF-2 target genes modestly in 786-O cells.Western Blot Analysis Cell Line:HEK293T cells Concentration:1 and 10?μM Incubation Time:Result:Reduced the physical association between HIF-2α and VHL.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    HIF/HIF Prolyl-hydroxylase
  • Recptor
    HIF-2α
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    874590-32-6
  • Formula Weight
    327.4
  • Molecular Formula
    C17H17N3O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:250 mg/mL?(763.59 mM)
  • SMILES
    O=S1(=O)N=C(Nc2ccccc2N2CCCC2)c2ccccc21
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Bidirectional Modulation of HIF-2 Activity through Chemical Ligands[C]// 中国生物化学与分子生物学会全国会员代表大会暨全国学术会议. 0.
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