IK-862

CAS No. 478911-60-3

IK-862( —— )

Catalog No. M34281 CAS No. 478911-60-3

IK-862 is a selective inhibitor of TACE (ADAM17).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 567 Get Quote
5MG 848 Get Quote
10MG 1159 Get Quote
25MG 1647 Get Quote
50MG 2254 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    IK-862
  • Note
    Research use only, not for human use.
  • Brief Description
    IK-862 is a selective inhibitor of TACE (ADAM17).
  • Description
    IK-862 is a selective inhibitor of TACE.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    MMP
  • Recptor
    MMP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    478911-60-3
  • Formula Weight
    433.5
  • Molecular Formula
    C25H27N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C[C@@]1(C(=O)N([C@@H](C(NO)=O)C)CC1)C2=CC=C(OCC=3C4=C(N=C(C)C3)C=CC=C4)C=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Georgiadis D, et al. Specific targeting of metzincin family members with small-molecule inhibitors: progress toward a multifarious challenge. Bioorg Med Chem. 2008;16(19):8781-8794. doi:10.1016/j.bmc.2008.08.058?
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